SCHEMBL28873199

SCHEMBL28873199

NCc1ccc(N)c(-c2cc[c]c(F)c2)c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 3/20 0.33
TAAR1 Q96RJ0 1/20 0.33
CSNK2A1 P68400 2/20 0.32
HRH3 Q9Y5N1 1/20 0.31
ROCK1 Q13464 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297202 0.78 TSHR (0.39)
SCHEMBL1244409 0.75
SCHEMBL28829313 0.71 DPP4 (0.52) TAAR1
SCHEMBL3790606 0.71 LOXL2 (0.54) LOXL2TAAR1CSNK2A1HRH3ROCK1
SCHEMBL3789650 0.71 CSNK2A1 (0.59) LOXL2TAAR1CSNK2A1HRH3ROCK1
SCHEMBL3790111 0.70 MAP4K4 (0.46) LOXL2TAAR1CSNK2A1HRH3
SCHEMBL27414053 0.69 LOXL2 (0.37) LOXL2TAAR1
SCHEMBL27784685 0.69 LOXL2 (0.37) LOXL2TAAR1
SCHEMBL7861005 0.69
SCHEMBL28297213 0.68 CYP3A4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN disclosed