SCHEMBL28297213

SCHEMBL28297213

Nc1cc(Cl)ccc1-c1cc[c]c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.39
ALDH1A1 P00352 4/20 0.39
TSHR P16473 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
ALOX15 P16050 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
TP53 P04637 1/20 0.38
HPGD P15428 2/20 0.36
ALOX12 P18054 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GRM5 P41594 1/20 0.34
KDM4E B2RXH2 2/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 1/20 0.33
CYP1A2 P05177 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP2C19 P33261 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297202 0.87 TSHR (0.39) CYP3A4ALDH1A1TSHRSMN1; SMN2ALOX15
SCHEMBL435211 0.83 AHR (0.48) ALDH1A1TSHRSMN1; SMN2TP53HPGD
SCHEMBL433433 0.83 GRM2 (0.36) AHR
SCHEMBL15622693 0.77 TSHR (0.46) CYP3A4ALDH1A1TSHRSMN1; SMN2ALOX15
SCHEMBL2500848 0.75 TSHR (0.45) CYP3A4ALDH1A1TSHRSMN1; SMN2ALOX15
SCHEMBL433164 0.74 ALOX5 (0.42) ALDH1A1TSHRSMN1; SMN2TP53HPGD
SCHEMBL14906969 0.73 ALDH1A1 (0.56) CYP3A4ALDH1A1TSHRSMN1; SMN2ALOX15
SCHEMBL17867987 0.73 TSHR (0.46) CYP3A4ALDH1A1TSHRSMN1; SMN2ALOX15
SCHEMBL4148009 0.73 SMN1; SMN2 (0.46) CYP3A4ALDH1A1TSHRSMN1; SMN2ALOX15
SCHEMBL17514779 0.72 NISCH (0.38) ALDH1A1SMN1; SMN2TP53HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109906220-A For treating the 1,3- dihydro -1,4- benzodiazepine * -2- thione compounds of CNS related disease 豪夫迈·罗氏有限公司 2019-06-18 CN disclosed