SCHEMBL28875987

SCHEMBL28875987

CC=CC(=O)Nc1ccc(-c2ccnc(Nc3ccccc3N3CCOCC3)n2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 20/20 0.76
JAK3 P52333 15/20 0.76
JAK1 P23458 9/20 0.76
TYK2 P29597 6/20 0.65
HDAC1 Q13547 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
HDAC3 O15379 1/20 0.50
NCOR1 O75376 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
IKBKB O14920 1/20 0.49
PDGFRB P09619 1/20 0.49
KIT P10721 1/20 0.49
PDGFRA P16234 1/20 0.49
FLT1 P17948 1/20 0.49
RPS6KB1 P23443 1/20 0.49
FLT4 P35916 1/20 0.49
KDR P35968 1/20 0.49
FLT3 P36888 1/20 0.49
MAP3K9 P80192 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28876006 0.91 JAK2 (0.77) JAK2JAK3JAK1TYK2
SCHEMBL28875997 0.89 JAK2 (0.75) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL29813618 0.86 JAK2 (1.00) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL28875980 0.86 JAK2 (1.00) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL28876016 0.82 JAK3 (0.76) JAK2JAK3JAK1TYK2FLT3
SCHEMBL17287879 0.81 JAK2 (0.56) JAK2JAK3JAK1TYK2HDAC1
SCHEMBL28876014 0.80 JAK3 (0.77) JAK2JAK3JAK1TYK2
SCHEMBL28556666 0.80 JAK2 (0.77) JAK2JAK3JAK1TYK2IKBKB
SCHEMBL29813581 0.79 JAK2 (1.00) JAK2JAK3JAK1TYK2
SCHEMBL28875975 0.79 JAK2 (1.00) JAK2JAK3JAK1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330484-B Substituted phenyl pyrimidine derivative as JAK kinase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application 中国药科大学 2022-08-26 CN disclosed