SCHEMBL28876014

SCHEMBL28876014

C=CC(=O)Nc1cccc(-c2ccnc(Nc3ccccc3N3CCOCC3)n2)c1

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 8/20 0.77
JAK2 O60674 7/20 0.77
JAK1 P23458 5/20 0.77
TYK2 P29597 4/20 0.77
EGFR P00533 4/20 0.56
BTK Q06187 6/20 0.55
ITK Q08881 1/20 0.51
SMG1 Q96Q15 1/20 0.51
SCN9A Q15858 1/20 0.51
CAMK2D Q13557 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28875997 0.90 JAK2 (0.75) JAK3JAK2JAK1TYK2EGFR
SCHEMBL28876006 0.90 JAK2 (0.77) JAK3JAK2JAK1TYK2SMG1
SCHEMBL28876009 0.87 JAK2 (1.00) JAK3JAK2JAK1TYK2EGFR
SCHEMBL29813541 0.87 JAK2 (1.00) JAK3JAK2JAK1TYK2EGFR
SCHEMBL15637731 0.86 JAK2 (0.80) JAK3JAK2JAK1TYK2EGFR
SCHEMBL17071413 0.86 JAK2 (0.88) JAK3JAK2JAK1TYK2EGFR
SCHEMBL17071335 0.86 JAK3 (0.79) JAK3JAK2JAK1TYK2EGFR
SCHEMBL17071334 0.86 JAK3 (0.79) JAK3JAK2JAK1TYK2EGFR
SCHEMBL17071342 0.84 JAK3 (0.75) JAK3JAK2JAK1TYK2EGFR
SCHEMBL28875996 0.83 JAK3 (0.76) JAK3JAK2JAK1TYK2BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330484-B Substituted phenyl pyrimidine derivative as JAK kinase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application 中国药科大学 2022-08-26 CN disclosed