SCHEMBL28876006

SCHEMBL28876006

CC=CC(=O)Nc1cccc(-c2ccnc(Nc3ccccc3N3CCOCC3)n2)c1

nearest known ligand 0.77

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 12/20 0.77
JAK3 P52333 7/20 0.77
TYK2 P29597 3/20 0.77
JAK1 P23458 6/20 0.62
SMG1 Q96Q15 3/20 0.49
SCN9A Q15858 2/20 0.49
CAMK2D Q13557 1/20 0.48
CDK1 P06493 1/20 0.48
CDK2 P24941 1/20 0.48
PLK1 P53350 1/20 0.47
MTOR P42345 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28875987 0.91 JAK2 (0.76) JAK2JAK3TYK2JAK1
SCHEMBL28876014 0.90 JAK3 (0.77) JAK2JAK3TYK2JAK1SMG1
SCHEMBL29813581 0.87 JAK2 (1.00) JAK2JAK3TYK2JAK1
SCHEMBL28875975 0.87 JAK2 (1.00) JAK2JAK3TYK2JAK1
SCHEMBL28875991 0.84 JAK3 (0.77) JAK2JAK3TYK2JAK1SCN9A
SCHEMBL28394053 0.84 JAK3 (0.55) JAK2JAK3TYK2JAK1SCN9A
SCHEMBL28387824 0.84 JAK3 (0.55) JAK2JAK3TYK2JAK1SCN9A
SCHEMBL28382437 0.81 JAK3 (0.52) JAK2JAK3TYK2JAK1SCN9A
SCHEMBL28383508 0.81 JAK3 (0.52) JAK2JAK3TYK2JAK1SCN9A
SCHEMBL28875997 0.80 JAK2 (0.75) JAK2JAK3TYK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110330484-B Substituted phenyl pyrimidine derivative as JAK kinase inhibitor or pharmaceutically acceptable salt thereof, preparation method and application 中国药科大学 2022-08-26 CN disclosed