SCHEMBL28876190

SCHEMBL28876190

COc1cc(NCCCl)cc(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 3/20 0.46
KMT2A Q03164 3/20 0.43
POLB P06746 1/20 0.43
PRKACA P17612 1/20 0.41
PRKACG P22612 1/20 0.41
PRKACB P22694 1/20 0.41
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
KDM4E B2RXH2 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11168082 0.88 MAPT (0.44) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL10989612 0.81 MTNR1A (0.60) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL12178218 0.81 KMT2A (0.48) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL27787646 0.79 TAAR1 (0.47) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL28572444 0.79 GAA (0.47) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL14788156 0.79 KMT2A (0.47) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL27848998 0.79 GAA (0.76) GAAMAPTALDH1A1KMT2AKDM4E
SCHEMBL10010025 0.78 POLB (0.46) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL11118508 0.76 KDR (0.45) GAAMAPTALDH1A1KMT2APOLB
SCHEMBL6900277 0.76 ALDH1A1 (0.52) GAAMAPTALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115108926-B Intermediate compound for preparing erdasatinib and preparation method 上海工程技术大学 2023-06-20 CN claimed
CN-115108926-A Intermediate compound for preparing erdastinib and preparation method 上海工程技术大学 2022-09-27 CN claimed
CN-115108926-B Intermediate compound for preparing erdasatinib and preparation method 上海工程技术大学 2023-06-20 CN disclosed
CN-115108926-B Intermediate compound for preparing erdasatinib and preparation method 上海工程技术大学 2023-06-20 CN disclosed
CN-115108926-A Intermediate compound for preparing erdastinib and preparation method 上海工程技术大学 2022-09-27 CN disclosed
CN-115108926-A Intermediate compound for preparing erdastinib and preparation method 上海工程技术大学 2022-09-27 CN disclosed