SCHEMBL28877321

SCHEMBL28877321

FC(F)=C(CBr)CCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.47
TDP1 Q9NUW8 3/20 0.46
ALDH1A1 P00352 4/20 0.44
FFAR1 O14842 2/20 0.44
HDAC2 Q92769 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC1 Q13547 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HDAC3 O15379 1/20 0.39
MAPK1 P28482 1/20 0.39
ADRA1A P35348 1/20 0.39
HDAC4 P56524 1/20 0.39
SLC6A3 Q01959 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
TSHR P16473 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8665089 0.78 KEAP1 (0.64) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL10049328 0.74 KEAP1 (0.54) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL4192449 0.73 KEAP1 (0.58) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL10049324 0.71 ALDH1A1 (0.57) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL191218 0.71 KEAP1 (0.61) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL16795814 0.71 TDP1 (0.50) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL1498978 0.70 KEAP1 (0.67) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL28200575 0.70 KEAP1 (0.54) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL10049325 0.69 KEAP1 (0.48) KEAP1TDP1ALDH1A1FFAR1HDAC2
SCHEMBL4192865 0.69 FFAR1 (0.60) KEAP1TDP1ALDH1A1FFAR1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118684548-A Method for selective gem-difluoroallylation of (hetero) aryl phenols or polypeptides 中国科学院上海有机化学研究所 2024-09-24 CN disclosed
CN-115260069-B 3, 3-difluoroallylium salt compound and preparation method and application thereof 中国科学院上海有机化学研究所 2023-10-27 CN disclosed
CN-115260069-A 3,3-difluoroallylonium salt compound and preparation method and application thereof 中国科学院上海有机化学研究所 2022-11-01 CN disclosed