SCHEMBL28877902

SCHEMBL28877902

Nc1nc(N)c(N)c(-c2ccc(OC(F)F)nc2)n1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 3/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CB P42338 1/20 0.34
PI4KA P42356 1/20 0.34
PIK3CG P48736 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
MTOR P42345 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
DHFR P00374 2/20 0.32
ADORA1 P30542 3/20 0.32
ADORA2A P29274 3/20 0.32
ATR Q13535 1/20 0.32
DAO P14920 1/20 0.32
ADORA2B P29275 1/20 0.31
PTGES O14684 4/20 0.31
F2RL3 Q96RI0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28877904 0.81 MGMT (0.40) MTORPDE4APDE4BPDE4CPDE4D
SCHEMBL29974131 0.81 MGMT (0.40) MTORPDE4APDE4BPDE4CPDE4D
SCHEMBL28957972 0.79 ADORA2A (0.47) PIK3CGDHFRADORA1ADORA2A
SCHEMBL16076591 0.71 PTGES (0.38) PDE4APDE4BPDE4CPDE4DADORA2B
SCHEMBL29939288 0.69 KDM4E (0.50) PIK3CAPIK3CDPIK3CBDAO
SCHEMBL557830 0.69 KDM4E (0.50) PIK3CAPIK3CDPIK3CBDAO
SCHEMBL30607712 0.67 DPP4 (0.40) PIK3CAPIK3CDPIK3CBPDE4APDE4B
SCHEMBL16463518 0.65 CSNK1A1 (0.61) PIK3CGMTORPDE4APDE4DDHFR
SCHEMBL25324910 0.64 MAT2A (0.37) PIK3CAPIK3CDPIK3CBPDE4APDE4B
SCHEMBL9158351 0.64 DAO (0.42) DAOPTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115141202-A Pyrimidopyrazinone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-04 CN disclosed