SCHEMBL28879128

SCHEMBL28879128

C[C@@H]1CNC[C@@H](c2ccc3cccc(C(F)(F)F)c3n2)C1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.45
CHRNA4 P43681 4/20 0.45
CHRNB4 P30926 2/20 0.35
CHRNA3 P32297 2/20 0.35
HTR2C P28335 5/20 0.34
HTR2A P28223 4/20 0.34
HTR2B P41595 4/20 0.34
NCF1 P14598 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
SSTR4 P31391 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19837031 1.00 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C
SCHEMBL28879111 1.00 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C
SCHEMBL29962079 1.00 CHRNB2 (0.45) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C
SCHEMBL7966941 0.79 HTR2C (0.51) HTR2CNCF1
SCHEMBL19837189 0.71 TLR7 (0.55) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C
SCHEMBL14921560 0.67 METAP2 (0.47) CHRNB2CHRNA4NCF1
SCHEMBL17300871 0.66 CHRNB4 (0.52) CHRNB2CHRNA4CHRNB4CHRNA3HTR2C
SCHEMBL30019238 0.64 METAP2 (0.55)
SCHEMBL3462719 0.64 AURKA (0.41) HTR2AHTR2B
SCHEMBL31382556 0.63 NCF1 (0.53) NCF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563075-B TLR7/8 antagonists and uses thereof 默克专利股份公司 2022-09-30 CN disclosed