SCHEMBL28881256

SCHEMBL28881256

N#Cc1cccc(-c2cncc(/C=N/O)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 7/20 0.45
GABRB3 P28472 7/20 0.45
GABRA5 P31644 7/20 0.45
GABRA3 P34903 7/20 0.45
GABRA1 P14867 1/20 0.45
NEK1 Q96PY6 1/20 0.44
IDO1 P14902 2/20 0.43
CLK4 Q9HAZ1 1/20 0.42
CYP11B2 P19099 3/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNA5 P30532 1/20 0.40
CHRNA4 P43681 1/20 0.40
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
CYP11B1 P15538 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28881260 1.00 GABRG2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL29987372 1.00 GABRG2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28881564 0.84 CYP11B2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28881566 0.84 CYP11B2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL29987911 0.84 CYP11B2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL29987290 0.81 GABRG2 (0.48) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28881250 0.81 GABRG2 (0.48) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL5117029 0.81 PTPN5 (0.47) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL5117035 0.81 PTPN5 (0.47) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL8307833 0.79 MKNK1 (0.44) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304591-A Bridged steroid synthetase inhibitor and preparation method and application thereof 广州中医药大学(广州中医药研究院) 2022-11-08 CN disclosed