SCHEMBL29987290

SCHEMBL29987290

N#Cc1cccc(-c2cncc(C=O)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 7/20 0.48
GABRB3 P28472 7/20 0.48
GABRA5 P31644 7/20 0.48
GABRA3 P34903 7/20 0.48
GABRA1 P14867 1/20 0.48
IDO1 P14902 2/20 0.47
CLK4 Q9HAZ1 1/20 0.45
NEK1 Q96PY6 1/20 0.43
CYP11B2 P19099 3/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA5 P30532 1/20 0.43
CHRNA4 P43681 1/20 0.43
CYP11B1 P15538 2/20 0.42
CYP17A1 P05093 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
BRD4 O60885 1/20 0.42
BRD2 P25440 1/20 0.42
XDH P47989 1/20 0.41
SLC22A12 Q96S37 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28881250 1.00 GABRG2 (0.48) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL16180558 0.88 CYP11B1 (0.49) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL15821011 0.84 TRIM24 (0.49) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL746371 0.83 CYP11B2 (0.49) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28881256 0.81 GABRG2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL28881260 0.81 GABRG2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL29987372 0.81 GABRG2 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL5849310 0.79 XDH (0.50) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL1476029 0.79 RAF1 (0.47)
SCHEMBL30345862 0.77 MKNK1 (0.47) CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115304591-B Bridged ring steroid synthetase inhibitor and preparation method and application thereof 广州中医药大学(广州中医药研究院) 2024-10-01 CN disclosed
CN-115304591-A Bridged steroid synthetase inhibitor and preparation method and application thereof 广州中医药大学(广州中医药研究院) 2022-11-08 CN disclosed