SCHEMBL28885488

SCHEMBL28885488

C=CC(=O)Nc1ccc(OC2CCOCC2)c(F)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 0.61
ITK Q08881 5/20 0.61
HRH3 Q9Y5N1 1/20 0.53
TBK1 Q9UHD2 1/20 0.50
KDR P35968 2/20 0.44
TGM2 P21980 1/20 0.43
CCNT1 O60563 1/20 0.43
CDK7 P50613 1/20 0.43
CDK9 P50750 1/20 0.43
CCNH P51946 1/20 0.43
MNAT1 P51948 1/20 0.43
BRAF P15056 1/20 0.42
EPHX2 P34913 2/20 0.42
DGAT1 O75907 1/20 0.41
SOAT1 P35610 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20209233 0.88 EGFR (0.52) EGFRITKHRH3KDRTGM2
SCHEMBL28376476 0.88 EGFR (0.58) EGFRITKHRH3KDRTGM2
SCHEMBL28376609 0.86 RORC (0.58) EGFRITKTBK1
SCHEMBL28426333 0.85 EGFR (0.49) EGFRITKHRH3KDRTGM2
SCHEMBL28439175 0.85 EGFR (0.49) EGFRITKHRH3KDRTGM2
SCHEMBL28371428 0.85 POLB (0.56) EGFRITKTBK1TGM2
SCHEMBL28372603 0.85 PDE4D (0.53) EGFRITKTBK1TGM2
SCHEMBL24968537 0.83 P2RX4 (0.51) EGFRITK
SCHEMBL28371190 0.80 TGM2 (0.54) EGFRHRH3TBK1TGM2
SCHEMBL28375853 0.78 PDE4D (0.54) EGFRITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110981876-B 8-substituted styrylxanthine derivatives and uses thereof 广东东阳光药业有限公司 2021-10-01 CN disclosed
CN-110981876-A 8-substituted styrylxanthine derivatives and uses thereof 广东东阳光药业有限公司 2020-04-10 CN disclosed