SCHEMBL28889170

SCHEMBL28889170

NC(=O)C(c1cccc(F)c1)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43
AURKA O14965 2/20 0.41
USP2 O75604 1/20 0.40
KMT2A Q03164 1/20 0.40
ADRB2 P07550 1/20 0.39
PNMT P11086 1/20 0.39
EPHX1 P07099 4/20 0.39
KCNN4 O15554 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
NR3C2 P08235 1/20 0.38
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
CES2 O00748 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29893770 1.00 HDAC4 (0.43) HDAC4HDAC7HDAC5AURKAUSP2
SCHEMBL24110333 0.87 TACR1 (0.45) AURKAADRB2PNMTEPHX1NOS3
SCHEMBL29893620 0.86 AURKA (0.40) AURKAADRB2PNMTEPHX1OPRL1
SCHEMBL28889316 0.86 AURKA (0.40) AURKAADRB2PNMTEPHX1OPRL1
SCHEMBL28889280 0.86 AURKA (0.40) AURKAADRB2PNMTEPHX1NR3C2
SCHEMBL29893670 0.86 AURKA (0.40) AURKAADRB2PNMTEPHX1NR3C2
SCHEMBL28889226 0.86 AURKA (0.42) AURKAKMT2AADRB2PNMTEPHX1
SCHEMBL29893797 0.86 AURKA (0.42) AURKAKMT2AADRB2PNMTEPHX1
SCHEMBL28889259 0.85 HDAC4 (0.42) HDAC4HDAC7HDAC5AURKAUSP2
SCHEMBL28889273 0.85 ADRB2 (0.40) AURKAKMT2AADRB2EPHX1KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed