SCHEMBL28889190

SCHEMBL28889190

CC(C)c1ccccc1C(C#N)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.40
TRPV3 Q8NET8 1/20 0.37
KCNN4 O15554 1/20 0.36
NOS3 P29474 1/20 0.36
NOS2 P35228 1/20 0.36
NPSR1 Q6W5P4 2/20 0.35
AR P10275 1/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
LRRK2 Q5S007 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
IDH2 P48735 1/20 0.34
POLB P06746 1/20 0.33
ALDH1A1 P00352 2/20 0.33
TAAR1 Q96RJ0 1/20 0.33
PKM P14618 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889210 0.87 ADRB2 (0.40) ADRB2TRPV3KCNN4NOS3NOS2
SCHEMBL28889282 0.85 ALDH1A1 (0.40) ADRB2TRPV3KCNN4NOS3NOS2
SCHEMBL28994023 0.85 KDM4E (0.41) ADRB2TRPV3NOS3NOS2AR
SCHEMBL28889203 0.84 ALDH1A1 (0.50) ADRB2TRPV3NOS3NOS2NPSR1
SCHEMBL28889153 0.83 ADRB2 (0.40) ADRB2TRPV3KCNN4NOS3NOS2
SCHEMBL28889197 0.82 ADRB2 (0.38) ADRB2TRPV3KCNN4NOS3NOS2
SCHEMBL24110401 0.81 ALDH1A1 (0.47) ADRB2TRPV3NOS3NOS2NPSR1
SCHEMBL28889345 0.81 ADRB2 (0.37) ADRB2TRPV3KCNN4NOS3NOS2
SCHEMBL28889369 0.80 ADRB2 (0.38) ADRB2TRPV3KCNN4NOS3NOS2
SCHEMBL28889321 0.77 ADRB2 (0.41) ADRB2TRPV3KCNN4NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed