SCHEMBL28889369

SCHEMBL28889369

COc1ncccc1C(C#N)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.38
KCNN4 O15554 1/20 0.36
NFE2L2 Q16236 3/20 0.36
MAT2A P31153 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPV3 Q8NET8 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
ATM Q13315 1/20 0.34
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
AHR P35869 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28994023 0.85 KDM4E (0.41) ADRB2KDM4EMEN1KMT2ATRPV3
SCHEMBL28889153 0.84 ADRB2 (0.40) ADRB2KCNN4KDM4ETRPV3ALDH1A1
SCHEMBL28889197 0.83 ADRB2 (0.38) ADRB2KCNN4KDM4ETRPV3ALDH1A1
SCHEMBL28889245 0.81 KDM4E (0.41) ADRB2KDM4EMEN1KMT2AATM
SCHEMBL28889210 0.80 ADRB2 (0.40) ADRB2KCNN4KDM4EMEN1KMT2A
SCHEMBL28889190 0.80 ADRB2 (0.40) ADRB2KCNN4MAT2AKDM4ETRPV3
SCHEMBL28889282 0.79 ALDH1A1 (0.40) ADRB2KCNN4KDM4EMEN1KMT2A
SCHEMBL28889203 0.78 ALDH1A1 (0.50) ADRB2KDM4ETRPV3ATMALDH1A1
SCHEMBL28889381 0.77 ADRB2 (0.39) ADRB2KCNN4NFE2L2MAT2ATRPV3
SCHEMBL28889345 0.77 ADRB2 (0.37) ADRB2KCNN4KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed