SCHEMBL28889348

SCHEMBL28889348

N#CC(c1cc(C(F)(F)F)ccn1)c1c(F)cccc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.42
ALDH1A1 P00352 2/20 0.42
ADRB2 P07550 1/20 0.39
NOS3 P29474 1/20 0.38
NOS2 P35228 1/20 0.38
CTSS P25774 1/20 0.36
LRRK2 Q5S007 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GPBAR1 Q8TDU6 3/20 0.35
KDM4E B2RXH2 3/20 0.34
PKM P14618 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KCNN4 O15554 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
ABL1 P00519 1/20 0.32
MAP2K2 P36507 1/20 0.32
CSNK1A1 P48729 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28889345 0.85 ADRB2 (0.37) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL28889282 0.85 ALDH1A1 (0.40) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL28889321 0.85 ADRB2 (0.41) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL28889353 0.81 GAA (0.44) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL29894681 0.81 GAA (0.44) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL28889240 0.81 ADRB2 (0.38) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL24110401 0.80 ALDH1A1 (0.47) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL30484313 0.79 L3MBTL1 (0.44) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL28889197 0.78 ADRB2 (0.38) GAAALDH1A1ADRB2NOS3NOS2
SCHEMBL28889258 0.78 ADRB2 (0.39) GAAALDH1A1ADRB2NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022222911-A1 PYRIMIDONE COMPOUND AND USE THEREOF 武汉人福创新药物研发中心有限公司 2022-10-27 WO disclosed
CN-115215862-A Pyrimidone compounds and uses thereof 武汉人福创新药物研发中心有限公司 2022-10-21 CN disclosed