SCHEMBL28889677

SCHEMBL28889677

Cn1nc(C(F)F)cc1NC(=O)c1cccc(F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.55
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
GRM5 P41594 1/20 0.50
MAPT P10636 3/20 0.49
CYP2C19 P33261 2/20 0.48
CYP1A2 P05177 1/20 0.48
TSHR P16473 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
ALOX15 P16050 1/20 0.47
KCNK3 O14649 2/20 0.47
KCNK9 Q9NPC2 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
TP53 P04637 3/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28398944 0.87 NPC1 (0.54) MEN1KMT2ASMN1; SMN2GRM5MAPT
SCHEMBL28400070 0.87 GAA (0.50) KDM4EMEN1KMT2AGRM5ALDH1A1
SCHEMBL28397870 0.86 GRM5 (0.49) SMN1; SMN2GRM5CYP2C19CYP1A2ALDH1A1
SCHEMBL30153272 0.86 GRM5 (0.49) SMN1; SMN2GRM5CYP2C19CYP1A2ALDH1A1
SCHEMBL28399770 0.85 LMNA (0.48) KDM4EMEN1KMT2ASMN1; SMN2GRM5
SCHEMBL28407311 0.84 TSHR (0.54) KDM4EMEN1KMT2ASMN1; SMN2GRM5
SCHEMBL28397875 0.84 LMNA (0.58) MEN1KMT2AMAPTTSHRGAA
SCHEMBL13056035 0.80 NQO2 (0.43) MEN1KMT2ASMN1; SMN2MAPTTSHR
SCHEMBL28398860 0.80 RAB9A (0.49) MEN1KMT2ASMN1; SMN2GRM5MAPT
SCHEMBL28401280 0.80 KDM4E (0.55) KDM4EMEN1KMT2ASMN1; SMN2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111187215-B Fluorine-containing pyrazole amide derivative, preparation method and application thereof 西北农林科技大学 2023-02-24 CN disclosed
CN-111187215-A Fluorine-containing pyrazole amide derivative, preparation method and application thereof 西北农林科技大学 2020-05-22 CN disclosed