SCHEMBL28890703

SCHEMBL28890703

COC(=O)c1ccc(COc2cccc(-c3ccc(OCC4CCOCC4)nc3)c2)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.43
GABRA5 P31644 6/20 0.42
CYP2D6 P10635 1/20 0.42
ACACA Q13085 2/20 0.41
PTGES O14684 3/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
GABRA1 P14867 1/20 0.39
SLC2A1 P11166 1/20 0.39
VDR P11473 1/20 0.39
F10 P00742 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28405014 0.94 ACACA (0.46) GABRA5ACACAPTGESMRGPRX4VDR
SCHEMBL20772827 0.93 FFAR4 (0.43) GABRA5ACACAPTGESMRGPRX4VDR
SCHEMBL20772768 0.91 PIM1 (0.43) PIM1GABRA5CYP2D6MRGPRX4
SCHEMBL20772999 0.88 SCN9A (0.44) PIM1GABRA5CYP2D6ACACAPTGES
SCHEMBL20772618 0.88 NR1H2 (0.46) PIM1GABRA5CYP2D6ACACAPTGES
SCHEMBL20772316 0.85 NR1H4 (0.48) ACACAPTGESMRGPRX4
SCHEMBL28410891 0.84 PTGES (0.45) GABRA5ACACAPTGESMRGPRX4
SCHEMBL20772628 0.84 PTGES (0.42) GABRA5ACACAPTGESMRGPRX4VDR
SCHEMBL20772603 0.84 ACACA (0.43) GABRA5ACACAPTGES
SCHEMBL28410957 0.84 VDR (0.42) GABRA5ACACAMRGPRX4VDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111132961-A Bisaryloxy derivatives as TTX-S blockers 拉夸里亚创药株式会社 2020-05-08 CN disclosed