SCHEMBL30002638

SCHEMBL30002638

COc1cc(F)c(N)cc1OCc1c(F)c(F)cc2cccnc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.41
CASP6 P55212 1/20 0.41
G6PD P11413 1/20 0.41
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
LMNA P02545 3/20 0.36
CYP1A2 P05177 2/20 0.36
ALDH1A1 P00352 2/20 0.36
PDE4A P27815 2/20 0.36
PDE4D Q08499 2/20 0.36
ABCB11 O95342 1/20 0.36
ESR1 P03372 1/20 0.36
PGR P06401 1/20 0.36
ADRB2 P07550 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRB1 P08588 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892621 1.00 NSD2 (0.41) NSD2CASP6G6PDPDGFRBPDGFRA
SCHEMBL30003250 0.87 NSD2 (0.41) NSD2CASP6G6PDPDGFRBPDGFRA
SCHEMBL28892537 0.87 NSD2 (0.41) NSD2CASP6G6PDPDGFRBPDGFRA
SCHEMBL28892170 0.82 KIT (0.36) NSD2CASP6G6PDSMN1; SMN2KIT
SCHEMBL30002605 0.82 KIT (0.36) NSD2CASP6G6PDSMN1; SMN2KIT
SCHEMBL30002047 0.82 ALDH1A1 (0.43) CASP6MEN1KMT2ANPC1RAB9A
SCHEMBL28892922 0.82 ALDH1A1 (0.43) CASP6MEN1KMT2ANPC1RAB9A
SCHEMBL30002712 0.81 NSD2 (0.47) NSD2CASP6G6PDPDGFRBPDGFRA
SCHEMBL28959473 0.81 NSD2 (0.47) NSD2CASP6G6PDPDGFRBPDGFRA
SCHEMBL28892522 0.79 MAOA (0.40) MEN1KMT2ACYP1A2MAOAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed