SCHEMBL28892256

SCHEMBL28892256

O=C1C=C(N(Cc2ccc(Cl)nc2)Cc2ccc(F)c(Cl)c2)CO1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.34
KCNQ2 O43526 1/20 0.34
KCNE1 P15382 1/20 0.34
KCNQ1 P51787 1/20 0.34
MDM2 Q00987 1/20 0.34
GRM2 Q14416 1/20 0.34
PARP1 P09874 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CTSL P07711 2/20 0.33
SLC6A9 P48067 2/20 0.32
KCNH2 Q12809 2/20 0.32
KDM1A O60341 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892266 0.92 MDM2 (0.34) KCNQ3KCNQ2KCNE1KCNQ1MDM2
SCHEMBL28892272 0.91 KCNQ3 (0.34) KCNQ3KCNQ2KCNE1KCNQ1MDM2
SCHEMBL28892391 0.90 CTSL (0.34) MDM2CTSLKDM1APSEN1PSEN2
SCHEMBL28892248 0.90 GBA1 (0.37) KCNH2
SCHEMBL28892338 0.89 IDO1 (0.34) MDM2GRM2PARP1CTSLKCNH2
SCHEMBL28892351 0.89 MDM2 (0.34) KCNQ3KCNQ2KCNE1KCNQ1MDM2
SCHEMBL28892262 0.88 OXTR (0.36) MDM2HDAC1HDAC6CTSLKDM1A
SCHEMBL28892406 0.88 HDAC1 (0.33) MDM2HDAC1HDAC6KDM1APSEN1
SCHEMBL28892369 0.87 LMNA (0.33) MDM2CTSLPSEN1PSEN2APH1B
SCHEMBL28892254 0.86 MDM2 (0.34) KCNQ3KCNQ2KCNE1KCNQ1MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558841-B 4- (N, N-disubstituted) furan-2 (5H) -ketone derivative, preparation method and application thereof 贵州大学 2022-04-12 CN disclosed