SCHEMBL2889408

SCHEMBL2889408

CCCc1c(I)nnn1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.50
ALDH1A1 P00352 5/20 0.46
ROCK1 Q13464 1/20 0.39
TP53 P04637 1/20 0.39
ALOX12 P18054 1/20 0.39
HTT P42858 1/20 0.38
USP2 O75604 1/20 0.38
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
NPC1 O15118 2/20 0.37
POLB P06746 1/20 0.37
MAPT P10636 2/20 0.36
CYP19A1 P11511 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2890539 0.79 MAOA (0.49) MAOAALDH1A1ROCK1TP53ALOX12
SCHEMBL17324731 0.75 HTT (0.51) MAOAALDH1A1ROCK1TP53ALOX12
SCHEMBL2885349 0.73 TP53 (0.46) ALDH1A1TP53ALOX12HTTSMN1; SMN2
SCHEMBL2891386 0.73 HTT (0.56) ALDH1A1TP53ALOX12HTTRAB9A
SCHEMBL29092087 0.72 SMN1; SMN2 (0.44) ALDH1A1TP53HTTRAB9ASMN1; SMN2
SCHEMBL17321500 0.72 ROCK1 (0.48) MAOAALDH1A1ROCK1TP53ALOX12
SCHEMBL15241806 0.69 ALDH1A1 (0.49) MAOAALDH1A1TP53ALOX12HTT
SCHEMBL4414691 0.69 HSD11B1 (0.57) ALDH1A1HTTSMN1; SMN2POLBMAPT
SCHEMBL12203848 0.68 ALDH1A1 (0.51) ALDH1A1RAB9APOLBMAPTGAA
SCHEMBL23399438 0.67 NR4A3 (0.53) ALDH1A1USP2RAB9APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858800-B2 Biaryl derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 2010-12-28 US disclosed
US-20070191389-A1 Biaryl derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-08-16 US disclosed
EP-1764362-A1 BIARYL DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-03-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070191389-A1 Biaryl derivatives GRM1, GRIN1, GRIN2B MAOA 1109/4885ALDH1A1 712/4885ROCK1 921/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.