SCHEMBL28895225

SCHEMBL28895225

NS(=O)(=O)Cc1ccc(Br)cn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.39
CA2 P00918 9/20 0.38
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
CA1 P00915 6/20 0.36
CA9 Q16790 6/20 0.36
CA5A P35218 2/20 0.36
ADRA2A P08913 2/20 0.35
ADRA2B P18089 2/20 0.35
ADRA2C P18825 2/20 0.35
PLAU P00749 1/20 0.35
GRM2 Q14416 1/20 0.35
CA12 O43570 2/20 0.34
LMNA P02545 1/20 0.34
MBOAT4 Q96T53 1/20 0.34
CA7 P43166 2/20 0.33
CA14 Q9ULX7 1/20 0.33
CA4 P22748 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9989117 0.81 GBA1 (0.43) GBA1CA2ALDH1A1KDM4ECA1
SCHEMBL15612266 0.78 GBA1 (0.37) GBA1CA2ALDH1A1KDM4EADRA2A
SCHEMBL16180689 0.78 GBA1 (0.41) GBA1ALDH1A1KDM4EGRM2LMNA
SCHEMBL29597062 0.77 NOS3 (0.42) CA2ALDH1A1KDM4ECA1CA9
SCHEMBL21827084 0.77 HTR2A (0.41) CA2CA1CA9CA5ACA12
SCHEMBL21826791 0.77 KDM4E (0.44) CA2KDM4ECA1CA9CA5A
SCHEMBL28649394 0.77 NOS3 (0.42) CA2ALDH1A1KDM4ECA1CA9
SCHEMBL31419110 0.77 GBA1 (0.40) GBA1ALDH1A1KDM4EGRM2LMNA
SCHEMBL1662137 0.77 GBA1 (0.40) GBA1ALDH1A1KDM4EGRM2LMNA
SCHEMBL21767155 0.74 APLNR (0.39) GBA1CA2ALDH1A1KDM4EADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111349043-B Intermediate for preparing pimenib and preparation method and application thereof 上海医药工业研究院 2022-09-27 CN disclosed
CN-111349043-A Intermediate for preparing pimenib and preparation method and application thereof 上海医药工业研究院 2020-06-30 CN disclosed