SCHEMBL3120908

SCHEMBL3120908

CC(=O)c1c(C)cc(NC(=O)OC(C)(C)C)cc1C

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA9 Q16790 1/20 0.48
CYP17A1 P05093 3/20 0.42
LCK P06239 2/20 0.39
PSMB8 P28062 1/20 0.39
NAMPT P43490 1/20 0.39
MAP4K4 O95819 1/20 0.39
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
KDM4E B2RXH2 1/20 0.37
EGLN2 Q96KS0 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
PPARG P37231 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16302366 0.87 CA12 (0.51) CA12CA1CA9CYP17A1LCK
SCHEMBL14439972 0.84 CA12 (0.49) CA12CA1CA9CYP17A1LCK
SCHEMBL9288893 0.83 CYP3A4 (0.47) CA12CA1CA9CYP17A1LCK
SCHEMBL849917 0.83 CA12 (0.48) CA12CA1CA9CYP17A1LCK
SCHEMBL25620110 0.83 CA12 (0.48) CA12CA1CA9CYP17A1LCK
SCHEMBL16991873 0.82 ALDH1A1 (0.49) CA12CA1CA9CYP17A1KDM4E
SCHEMBL28895283 0.82 CA12 (0.42) CA12CA1CA9CYP17A1LCK
SCHEMBL31206290 0.82 CA12 (0.42) CA12CA1CA9CYP17A1LCK
SCHEMBL28895279 0.81 CA12 (0.41) CA12CA1CA9CYP17A1LCK
SCHEMBL7477384 0.80 CA12 (0.48) CA12CA1CA9CYP17A1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001220-A1 NEW 1,2,4-TRIAZINE DERIVATIVES AND BIOLOGICAL APPLICATIONS THEREOF MUTABILIS SA (FR) 2010-01-07 WO disclosed
EP-2141164-A1 New 1,2,4-triazine derivatives and biological applications thereof Mutabilis (FR) 2010-01-06 EP disclosed