SCHEMBL28895492

SCHEMBL28895492

COC(=O)c1ncn(Cc2ccc(Cl)cc2)c1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.58
TSHR P16473 2/20 0.58
GAA P10253 2/20 0.58
SCD O00767 1/20 0.48
CYP11B2 P19099 2/20 0.45
CYP11B1 P15538 1/20 0.45
HSP90AA1 P07900 1/20 0.43
HSP90B1 P14625 1/20 0.43
YTHDC1 Q96MU7 1/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NR3C1 P04150 1/20 0.41
DRD2 P14416 1/20 0.41
TBXA2R P21731 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20591090 0.92 SCD (0.50) PKMTSHRGAASCDCYP11B2
SCHEMBL28441306 0.90 PKM (0.58) PKMTSHRGAASCDCYP11B2
SCHEMBL4150358 0.89 PKM (0.74) PKMTSHRGAACYP11B2CYP11B1
SCHEMBL28150125 0.88 PKM (0.57) PKMTSHRGAACYP11B2CYP11B1
SCHEMBL28430515 0.88 PKM (0.57) PKMTSHRGAACYP11B2CYP11B1
SCHEMBL28441301 0.88 PKM (0.53) PKMTSHRGAASCDSMN1; SMN2
SCHEMBL28436553 0.87 PKM (0.59) PKMTSHRGAAYTHDC1KMT2A
SCHEMBL7009864 0.86 YTHDC1 (0.46) PKMTSHRGAASCDCYP11B2
SCHEMBL20591091 0.86 SCD (0.46) PKMTSHRGAASCDCYP11B2
SCHEMBL28151121 0.86 PKM (0.54) PKMTSHRGAACYP11B2YTHDC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106692138-B Application of N-benzyl imidazole amide derivative as polymyxin antibiotic synergist 广州英赛特生物技术有限公司 2020-08-04 CN disclosed