SCHEMBL7009864

SCHEMBL7009864

COC(=O)c1ncn(Cc2ccc(C(=O)c3ccc(Cl)cc3)cc2)c1C(=O)OC

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.46
SCD O00767 1/20 0.46
VNN1 O95497 2/20 0.45
DRD2 P14416 3/20 0.43
TBXA2R P21731 3/20 0.43
CYP11B2 P19099 2/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP11B1 P15538 1/20 0.43
PKM P14618 2/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90B1 P14625 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20591090 0.94 SCD (0.50) YTHDC1SCDDRD2TBXA2RCYP11B2
SCHEMBL20591091 0.88 SCD (0.46) YTHDC1SCDCYP11B2RAB9AMEN1
SCHEMBL28895492 0.86 PKM (0.58) YTHDC1SCDDRD2TBXA2RCYP11B2
SCHEMBL20591084 0.83 PKM (0.47) YTHDC1SCDCYP11B2RAB9AKMT2A
SCHEMBL20591093 0.82 CYP11B2 (0.48) CYP11B2MEN1KMT2ACYP11B1PKM
SCHEMBL20591088 0.82 CYP11B2 (0.48) YTHDC1CYP11B2MEN1KMT2ACYP11B1
SCHEMBL4150352 0.82 PKM (0.62) CYP11B2CYP11B1PKMGAATSHR
SCHEMBL20591094 0.81 NOTUM (0.49) YTHDC1SCDPKMGAATSHR
SCHEMBL20591078 0.81 GAA (0.48) YTHDC1KMT2APKMGAATSHR
SCHEMBL20591075 0.80 MAPK8 (0.48) YTHDC1CYP11B2PKMGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed