SCHEMBL28895772

SCHEMBL28895772

CC(C)Oc1cc2c(cc1[N+](=O)[O-])CCCCN2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
ALDH1A1 P00352 1/20 0.44
PDK1 Q15118 1/20 0.39
XDH P47989 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A4 P31645 1/20 0.33
DRD3 P35462 1/20 0.33
OPRK1 P41145 1/20 0.33
HTR2B P41595 1/20 0.33
GFER P55789 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
MAPK1 P28482 2/20 0.32
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
ATM Q13315 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11518151 0.91 MAPT (0.54) MAPTALDH1A1PDK1XDHCYP1A2
SCHEMBL15283631 0.81 PDK1 (0.38) MAPTPDK1XDHCYP1A2CYP2D6
SCHEMBL6221710 0.80 ALDH1A1 (0.50) MAPTALDH1A1TDP1KMT2AMEN1
Hydrochloric Acid SCHEMBL9331091 0.79 ALDH1A1 (0.49) MAPTALDH1A1TDP1KMT2AMEN1
SCHEMBL28437849 0.77 CYP1A2 (0.37) MAPTPDK1XDHCYP1A2CYP2D6
SCHEMBL2205120 0.76 ALDH1A1 (0.51) MAPTALDH1A1CA12CA1CA2
SCHEMBL29581365 0.75 ALDH1A1 (0.57) MAPTALDH1A1TDP1KMT2AMEN1
SCHEMBL2205220 0.75 ALDH1A1 (0.57) MAPTALDH1A1TDP1KMT2AMEN1
SCHEMBL28374884 0.75 PDK1 (0.46) MAPTPDK1XDHSLC6A4HTR2B
SCHEMBL2206732 0.73 MAPT (0.48) MAPTALDH1A1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107652303-B Novel thienopyrimidine derivatives, preparation method and therapeutic use thereof 赛诺菲 2020-08-04 CN disclosed