SCHEMBL28895891

SCHEMBL28895891

COc1cccc(C2=CC=CC(N)C2(C)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.43
KDM1B Q8NB78 2/20 0.39
DYRK1A Q13627 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
BACE1 P56817 5/20 0.37
KCNH2 Q12809 3/20 0.37
MAOB P27338 2/20 0.37
NOTUM Q6P988 1/20 0.37
NCOA1 Q15788 1/20 0.36
NCOA3 Q9Y6Q9 1/20 0.36
KDM4E B2RXH2 1/20 0.36
KMT2A Q03164 1/20 0.36
PGR P06401 1/20 0.36
CYP3A4 P08684 2/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2E1 P05181 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28959780 0.82 KDM1A (0.40) KDM1AKDM1BDYRK1ACLK4MAOB
SCHEMBL20610266 0.76 PGR (0.41) DYRK1ACLK4BACE1KCNH2MAOB
SCHEMBL28646266 0.71 DYRK1A (0.50) KDM1ADYRK1ACLK4MAOBNOTUM
SCHEMBL196765 0.66 CYP3A4 (0.73) DYRK1ACLK4MAOBNOTUMKDM4E
SCHEMBL29489425 0.66 CYP3A4 (0.73) DYRK1ACLK4MAOBNOTUMKDM4E
Hydrogen Sulfide SCHEMBL28640169 0.64 CYP3A4 (0.70) DYRK1ACLK4MAOBNOTUMKDM4E
SCHEMBL29628977 0.64 CYP3A4 (0.77) DYRK1ACLK4MAOBNOTUMCYP3A4
Ammonia Solution, Strong SCHEMBL27960505 0.64 CYP3A4 (0.70) DYRK1ACLK4MAOBNOTUMKDM4E
SCHEMBL15624598 0.64 NFE2L2 (0.59) DYRK1ACLK4MAOBKDM4ECYP3A4
SCHEMBL1180343 0.62 ABL1 (0.69) DYRK1ACLK4MAOBCYP3A4CYP1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109890819-B Heterocyclic compounds as immunomodulators 因赛特公司 2022-11-22 CN disclosed