SCHEMBL28898102

SCHEMBL28898102

NC(=O)c1[nH]nc2c1COc1ccccc1-2

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 2/20 0.78
KDM4E B2RXH2 2/20 0.78
ALDH1A1 P00352 2/20 0.78
HSD17B10 Q99714 1/20 0.78
CCNA2 P20248 2/20 0.49
CDK2 P24941 2/20 0.49
CCNA1 P78396 2/20 0.49
THRB P10828 1/20 0.41
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
GSR P00390 2/20 0.39
KMT2A Q03164 2/20 0.39
AURKA O14965 1/20 0.39
PLK1 P53350 1/20 0.39
MAOB P27338 6/20 0.39
PIK3CD O00329 1/20 0.37
PIK3R2 O00459 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL646283 0.87 KDM4E (1.00) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL13539296 0.86 ALPL (0.78) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL13542004 0.83 ALDH1A1 (0.72) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL13539297 0.81 ALPL (1.00) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL13539303 0.80 ALDH1A1 (0.67) ALPLKDM4EALDH1A1HSD17B10RAB9A
SCHEMBL30759606 0.78 GSR (0.58) ALPLKDM4EALDH1A1HSD17B10CCNA2
SCHEMBL30290797 0.75 KDM4E (0.51) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL10176736 0.75 ALPL (0.61) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL4149139 0.72 ALPL (0.67) ALPLKDM4EALDH1A1HSD17B10THRB
SCHEMBL2171482 0.68 KDM4E (0.59) ALPLKDM4EALDH1A1HSD17B10THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531721-B Fused tricyclic pyrazole derivatives for modulating farnesoid X receptors 诺华股份有限公司 2020-07-17 CN claimed
CN-107531721-B Fused tricyclic pyrazole derivatives for modulating farnesoid X receptors 诺华股份有限公司 2020-07-17 CN disclosed