SCHEMBL28899162

SCHEMBL28899162

COc1ccc(Cn2ncc3ccc(N)cc3c2=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 12/20 0.56
AURKA O14965 1/20 0.53
GRK2 P25098 1/20 0.53
ROCK1 Q13464 1/20 0.53
RPS6KA1 Q15418 1/20 0.53
MCHR1 Q99705 1/20 0.52
PKM P14618 1/20 0.49
PKLR P30613 1/20 0.49
BRD4 O60885 1/20 0.48
PDE1A P54750 3/20 0.48
PDE1B Q01064 3/20 0.48
PDE1C Q14123 3/20 0.48
TDP1 Q9NUW8 1/20 0.48
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30579886 0.83 TDP1 (0.64) NPBWR1MCHR1PKMTDP1ALDH1A1
SCHEMBL5863967 0.83 TDP1 (0.56) AURKAGRK2ROCK1RPS6KA1PKM
SCHEMBL28899217 0.82 MAPT (0.52) NPBWR1AURKAGRK2ROCK1RPS6KA1
SCHEMBL20401464 0.81 QPCT (0.48) NPBWR1AURKAMCHR1BRD4PDE1A
SCHEMBL29447767 0.81 QPCT (0.48) NPBWR1AURKAMCHR1BRD4PDE1A
SCHEMBL22226011 0.80 NPBWR1 (0.62) NPBWR1AURKAGRK2ROCK1RPS6KA1
SCHEMBL25432622 0.79 NPBWR1 (0.55) NPBWR1MCHR1PKMPKLRPDE1A
SCHEMBL31513500 0.79 NPBWR1 (0.55) NPBWR1MCHR1PKMPKLRPDE1A
SCHEMBL4679664 0.76 NPBWR1 (0.61) NPBWR1MCHR1PKMPKLRPDE1A
SCHEMBL25431853 0.76 NPBWR1 (0.52) NPBWR1MCHR1PKMPKLRBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed