SCHEMBL28899217

SCHEMBL28899217

COc1ccc(Cn2ncc3ccc([N+](=O)[O-])cc3c2=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
NPBWR1 P48145 7/20 0.51
AURKA O14965 1/20 0.48
GRK2 P25098 1/20 0.48
ROCK1 Q13464 1/20 0.48
RPS6KA1 Q15418 1/20 0.48
MCL1 Q07820 1/20 0.47
MCHR1 Q99705 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CNR2 P34972 1/20 0.46
KAT2B Q92831 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5863497 0.85 TDP1 (0.51) MEN1KMT2ACNR2KAT2B
SCHEMBL20401101 0.83 GLS (0.57) MAPTSMN1; SMN2NPBWR1MEN1KMT2A
SCHEMBL28899162 0.82 NPBWR1 (0.56) NPBWR1AURKAGRK2ROCK1RPS6KA1
SCHEMBL5864274 0.79 PDE5A (0.43) MAPTSMN1; SMN2MEN1KMT2AKAT2B
SCHEMBL9874375 0.78 GLS (0.50) MAPTMEN1KMT2AKAT2B
SCHEMBL30579886 0.78 TDP1 (0.64) NPBWR1MCHR1
SCHEMBL30879415 0.77 DCTPP1 (0.45) MAPTSMN1; SMN2NPBWR1MCHR1MEN1
SCHEMBL22226011 0.75 NPBWR1 (0.62) MAPTNPBWR1AURKAGRK2ROCK1
SCHEMBL1163283 0.75 CNR2 (0.56) MAPTSMN1; SMN2CNR2
SCHEMBL25432622 0.74 NPBWR1 (0.55) NPBWR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109456308-B Heterocyclic compounds as ASK inhibitors and their use 南京圣和药业股份有限公司 2022-11-29 CN disclosed
CN-109456308-A Heterocyclic compound and its application as ASK inhibitor 南京圣和药业股份有限公司 2019-03-12 CN disclosed