SCHEMBL28900366

SCHEMBL28900366

COC(=O)c1ccc(-c2ccc3nc(SCC(OC)OC)ccc3c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.43
PDE7A Q13946 1/20 0.41
PDE7B Q9NP56 1/20 0.41
EGFR P00533 1/20 0.41
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
CYP19A1 P11511 1/20 0.40
MAPT P10636 6/20 0.40
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 5/20 0.40
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 1/20 0.40
RECQL P46063 1/20 0.40
CYP1A2 P05177 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22534223 0.82 KDM4E (0.42) KDM4EALDH1A1GAAMEN1KMT2A
SCHEMBL29935495 0.82 HDAC2 (0.42) CYP11B1CYP11B2MAPTKDM4EALDH1A1
SCHEMBL22534224 0.82 HDAC2 (0.42) CYP11B1CYP11B2MAPTKDM4EALDH1A1
SCHEMBL22534230 0.79 HRH3 (0.41)
SCHEMBL29935413 0.79 HRH3 (0.41)
SCHEMBL22534248 0.79 BACE1 (0.36) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL29935469 0.79 BACE1 (0.36) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL28476341 0.78 ALOX15 (0.42) ERN1PDE7APDE7BEGFRCYP11B1
SCHEMBL22534293 0.76 CYP1A2 (0.39) PDE7APDE7BKDM4EALDH1A1GAA
SCHEMBL22534239 0.76 RAB9A (0.40) MAPTKDM4EALDH1A1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111793025-B Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2022-09-23 CN disclosed
CN-111793025-A Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2020-10-20 CN disclosed