SCHEMBL28476341

SCHEMBL28476341

COC(=O)c1ccc(-c2ccc3nc(OCC(OC)OC)ccc3c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.42
HTT P42858 1/20 0.42
ERN1 O75460 1/20 0.41
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
CYP19A1 P11511 1/20 0.41
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.40
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40
RECQL P46063 1/20 0.40
HPGD P15428 2/20 0.40
NPC1 O15118 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10365973 0.82 ERN1 (0.49) ALOX15HTTERN1CYP11B1CYP11B2
SCHEMBL29935519 0.82 HDAC2 (0.43) CYP11B1CYP11B2ALDH1A1KDM4EMAPT
SCHEMBL22534298 0.82 HDAC2 (0.43) CYP11B1CYP11B2ALDH1A1KDM4EMAPT
SCHEMBL28470805 0.79 SCN9A (0.39)
SCHEMBL28901020 0.79 HRH3 (0.43) ALDH1A1HPGD
SCHEMBL28900366 0.78 ERN1 (0.43) ALOX15HTTERN1CYP11B1CYP11B2
SCHEMBL22534209 0.76 RXRA (0.38) ALDH1A1KDM4EMAPTPOLBNPC1
SCHEMBL22534222 0.74 CYP11B1 (0.37) CYP11B1CYP11B2GAAPDGFRBPDGFRA
SCHEMBL29935497 0.73 HTR3A (0.38) ALOX15HTTALDH1A1MAPTHPGD
SCHEMBL18617254 0.71 HTT (0.52) ALOX15HTTCYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111793025-B Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2022-09-23 CN disclosed
CN-111793025-A Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2020-10-20 CN disclosed