SCHEMBL28901020

SCHEMBL28901020

COC(COc1ccc2cc(-c3ccc(C#N)cc3)ccc2n1)OC

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.43
SCN7A Q01118 7/20 0.42
KCNH2 Q12809 5/20 0.41
MAP4K4 O95819 1/20 0.38
SCN10A Q9Y5Y9 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HPGDS O60760 1/20 0.36
PGR P06401 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22534298 0.84 HDAC2 (0.43) MAP4K4ALDH1A1
SCHEMBL29935519 0.84 HDAC2 (0.43) MAP4K4ALDH1A1
SCHEMBL28470805 0.81 SCN9A (0.39) SCN7AKCNH2SCN10A
SCHEMBL28476341 0.79 ALOX15 (0.42) ALDH1A1HPGD
SCHEMBL22534230 0.77 HRH3 (0.41) HRH3SCN10APGR
SCHEMBL29935413 0.77 HRH3 (0.41) HRH3SCN10APGR
SCHEMBL22534222 0.76 CYP11B1 (0.37)
SCHEMBL29935557 0.76 CYP11B1 (0.37)
SCHEMBL29935497 0.75 HTR3A (0.38) HRH3ALDH1A1HPGD
SCHEMBL2744804 0.71 MEN1 (0.49) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111793025-B Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2022-09-23 CN disclosed
CN-111793025-A Method for modifying amino in molecule by oxazoline quaternary ammonium salt and application thereof 中国科学院上海药物研究所 2020-10-20 CN disclosed