SCHEMBL28905979

SCHEMBL28905979

CS(=O)(=O)O.O=C(O)c1cccc(Br)n1

nearest known ligand 0.55

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
ALOX15 P16050 1/20 0.55
TSHR P16473 1/20 0.55
ACMSD Q8TDX5 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
GRM5 P41594 1/20 0.49
LMNA P02545 1/20 0.49
MMP2 P08253 1/20 0.48
CA1 P00915 6/20 0.45
CA2 P00918 6/20 0.45
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.41
ECE1 P42892 1/20 0.41
CTSA P10619 1/20 0.40
GNE Q9Y223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4989 0.89 KDM4E (0.70) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL29940784 0.89 KDM4E (0.70) KDM4EALOX15TSHRACMSDTDP1
Acetic Acid SCHEMBL28860398 0.87 KDM4E (0.61) KDM4EALOX15TSHRACMSDTDP1
Hydrochloric Acid SCHEMBL4538345 0.87 KDM4E (0.67) KDM4EALOX15TSHRACMSDTDP1
Acetamide SCHEMBL28213479 0.84 KDM4E (0.57) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL27924429 0.83 KDM4E (0.47) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL248932 0.79 GRM5 (0.54) ALDH1A1HPGDGRM5PTGS1PTGS2
SCHEMBL17258354 0.78 KDM4E (0.59) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL21245300 0.77 GRM5 (0.44) KDM4EALOX15TSHRACMSDTDP1
SCHEMBL28905985 0.76 GRM5 (0.43) KDM4EALOX15TSHRACMSDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115417814-A Synthetic method of 2-bromo-6-cyanopyridine 安徽大学 2022-12-02 CN claimed
CN-115417814-A Synthetic method of 2-bromo-6-cyanopyridine 安徽大学 2022-12-02 CN disclosed