SCHEMBL28906234

SCHEMBL28906234

Cc1cc(-c2cc(I)c[nH]2)cc(C)c1N1CCN(C)CC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.32
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDO2 P48775 1/20 0.30
MAP4K1 Q92918 1/20 0.30
ACHE P22303 1/20 0.30
TNKS O95271 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28513508 0.82 HRH4 (0.33) HRH4ALDH1A1POLBMAPTHTT
SCHEMBL28507573 0.82 MAP4K1 (0.40) HRH4ALDH1A1POLBMAPTHTT
SCHEMBL28507701 0.82 MAP4K1 (0.39) ALDH1A1MAPTSMN1; SMN2MAP4K1ACHE
SCHEMBL28502342 0.79 POLB (0.37) HRH4ALDH1A1POLBMAPTTNKS
SCHEMBL28517181 0.78 MELK (0.49) ALDH1A1MAPTHTTSMN1; SMN2MAP4K1
SCHEMBL20180762 0.77 MAPT (0.39) HRH4ALDH1A1POLBMAPTHTT
SCHEMBL28504472 0.73 MAPK13 (0.33) HRH4POLBMAPTTDO2
SCHEMBL28510220 0.72 KDM4E (0.43) HRH4ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL28506495 0.70 DRD2 (0.47) ALDH1A1POLBMAPTSMN1; SMN2MAP4K1
SCHEMBL28510206 0.70 WDR5 (0.39) POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed