SCHEMBL28906249

SCHEMBL28906249

COc1ccc(CN(CCO)C(=O)c2[nH]nc3ccc(Br)cc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.46
KDM4E B2RXH2 2/20 0.46
LMNA P02545 1/20 0.46
RECQL P46063 1/20 0.46
POLB P06746 2/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
SLC2A1 P11166 2/20 0.39
MMP1 P03956 1/20 0.39
MMP9 P14780 1/20 0.39
MMP13 P45452 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
PIK3R1 P27986 1/20 0.38
PIK3CA P42336 1/20 0.38
ALDH1A1 P00352 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LPAR1 Q92633 2/20 0.37
USP2 O75604 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16013442 0.75 KDM4E (0.51) TSHRKDM4ELMNARECQLPOLB
SCHEMBL21333004 0.70 TSHR (0.46) TSHRKDM4ELMNARECQLPOLB
SCHEMBL30285637 0.70 TSHR (0.46) TSHRKDM4ELMNARECQLPOLB
SCHEMBL3614141 0.70 TDP1 (0.54) TSHRPOLBMAPTGAAALDH1A1
SCHEMBL22413013 0.69 POLB (0.41) TSHRKDM4ELMNARECQLPOLB
SCHEMBL29863299 0.69 POLB (0.41) TSHRKDM4ELMNARECQLPOLB
SCHEMBL13547186 0.68 ALDH1A1 (0.49) TSHRKDM4ELMNARECQLPOLB
SCHEMBL28853322 0.67 LPAR1 (0.56) TSHRKDM4ELMNARECQLPOLB
SCHEMBL30301453 0.67 PRKACA (0.44) TSHRMAPTSLC2A1PIK3R1PIK3CA
SCHEMBL13319148 0.67 TSPO (0.51) TSHRKDM4EPOLBMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115433211-A Pyrazidopyridone methionine adenosyltransferase 2A inhibitors 南京正大天晴制药有限公司 2022-12-06 CN disclosed