SCHEMBL28906398

SCHEMBL28906398

Nc1cc(Cl)c(C2CC2)c(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.37
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31243002 1.00 CYP3A4 (0.39) CYP3A4ALDH1A1GAAMAPTTHRB
SCHEMBL15544603 0.85 CYP3A4 (0.48) CYP3A4ALDH1A1GAATHRBTSHR
SCHEMBL23043132 0.76 HSD17B10 (0.39) CYP3A4HTT
SCHEMBL25533309 0.76 KMT2A (0.35) ALDH1A1GAA
SCHEMBL23174552 0.76 GAA (0.39) GAAMAPT
SCHEMBL29679938 0.76 HSD17B10 (0.39) CYP3A4HTT
SCHEMBL28920148 0.73 MAPT (0.37) ALDH1A1GAAMAPTHTT
SCHEMBL26207348 0.73 MAOA (0.37) ALDH1A1
SCHEMBL3823135 0.73 KDM1A (0.38) CYP3A4ALDH1A1
SCHEMBL31527534 0.72 ALDH1A1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4713330-A1 TRICYCLIC COMPOUNDS AND USES THEREOF HUTCHMED Limited (CN) 2026-03-25 EP disclosed
WO-2024235286-A1 TRICYCLIC COMPOUNDS AND USES THEREOF HUTCHMED LIMITED (CN) 2024-11-21 WO disclosed
CN-115490709-A KRASG12D inhibitor and application thereof in medicine 四川海思科制药有限公司 2022-12-20 CN disclosed
CN-115304623-A Pyrimido-cyclic derivative and application thereof in medicine 四川海思科制药有限公司 2022-11-08 CN disclosed