SCHEMBL28909129

SCHEMBL28909129

CC(C)(NS(C)(=O)=O)c1cc(C(O)(C(N)F)C(F)F)nc(-c2ccc(F)cc2)c1Cl

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.34
PTGS2 P35354 7/20 0.34
MAPK14 Q16539 5/20 0.33
CYP3A4 P08684 3/20 0.33
CFTR P13569 3/20 0.33
SCN9A Q15858 1/20 0.31
KIT P10721 1/20 0.31
RXRA P19793 1/20 0.31
NR1H2 P55055 1/20 0.31
NR1H3 Q13133 1/20 0.31
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958770 0.82 CFTR (0.37) TRPV1PTGS2CFTRSCN9APTGS1
SCHEMBL25686557 0.82 CFTR (0.37) TRPV1PTGS2CFTRSCN9APTGS1
SCHEMBL23958851 0.82 CFTR (0.37) TRPV1PTGS2CFTRSCN9APTGS1
SCHEMBL30007267 0.80 PTGS2 (0.38) PTGS2SCN9AKITPTGS1
SCHEMBL23958629 0.80 PTGS2 (0.38) PTGS2SCN9AKITPTGS1
SCHEMBL23958600 0.75 CFTR (0.36) TRPV1PTGS2MAPK14CYP3A4CFTR
SCHEMBL28909197 0.75 CFTR (0.36) PTGS2MAPK14CFTRSCN9APTGS1
SCHEMBL23958691 0.75 CFTR (0.38) TRPV1PTGS2MAPK14CFTRSCN9A
SCHEMBL23958852 0.74 CFTR (0.35) TRPV1PTGS2MAPK14CYP3A4CFTR
SCHEMBL23958624 0.72 PTGS2 (0.36) PTGS2MAPK14SCN9AKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115461336-A RSV inhibiting 3-substituted quinoline and cinnoline derivatives 爱尔兰詹森科学公司 2022-12-09 CN disclosed