SCHEMBL23958852

SCHEMBL23958852

CC(C)(NS(C)(=O)=O)c1cc(C(CN)C(F)(F)F)nc(-c2ccc(F)cc2)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.35
PTGS2 P35354 9/20 0.32
CYP3A4 P08684 1/20 0.32
MAPK14 Q16539 1/20 0.32
SCN9A Q15858 1/20 0.31
TRPV1 Q8NER1 2/20 0.31
PTGS1 P23219 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MITF O75030 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
STAT3 P40763 1/20 0.31
STAT1 P42224 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TLR9 Q9NR96 1/20 0.31
KIT P10721 1/20 0.31
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958593 0.82 CFTR (0.39) CFTRSMN1; SMN2ADORA2AADORA1
SCHEMBL30007267 0.80 PTGS2 (0.38) PTGS2SCN9APTGS1KDM4EMITF
SCHEMBL23958629 0.80 PTGS2 (0.38) PTGS2SCN9APTGS1KDM4EMITF
SCHEMBL23958770 0.78 CFTR (0.37) CFTRPTGS2SCN9ATRPV1PTGS1
SCHEMBL25686557 0.78 CFTR (0.37) CFTRPTGS2SCN9ATRPV1PTGS1
SCHEMBL23958851 0.78 CFTR (0.37) CFTRPTGS2SCN9ATRPV1PTGS1
SCHEMBL23958600 0.75 CFTR (0.36) CFTRPTGS2CYP3A4MAPK14SCN9A
SCHEMBL28909129 0.74 TRPV1 (0.34) CFTRPTGS2CYP3A4MAPK14SCN9A
SCHEMBL23958763 0.73 CFTR (0.40) CFTRSCN9AKDM4EALDH1A1LMNA
SCHEMBL23958626 0.73 CFTR (0.40) CFTRSCN9AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed