SCHEMBL28922124

SCHEMBL28922124

NS(=O)(=O)c1cnc(OCCC2CCCOC2)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATXN2 Q99700 2/20 0.40
FFAR2 O15552 1/20 0.37
BRD4 O60885 2/20 0.36
ALDH1A1 P00352 1/20 0.35
CDK2 P24941 9/20 0.35
CDK1 P06493 7/20 0.35
CCNB1 P14635 5/20 0.35
CCNT1 O60563 4/20 0.35
CDK7 P50613 4/20 0.35
CDK9 P50750 4/20 0.35
CCNH P51946 4/20 0.35
CDK5 Q00535 4/20 0.35
CCNA2 P20248 5/20 0.34
CCNA1 P78396 5/20 0.34
CCNB2 O95067 2/20 0.33
CCNB3 Q8WWL7 2/20 0.33
NEK2 P51955 1/20 0.33
ROCK2 O75116 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1700291 0.86 ATXN2 (0.37) ATXN2FFAR2BRD4ALDH1A1
SCHEMBL28634010 0.86 ATXN2 (0.39) ATXN2FFAR2BRD4CDK2CDK1
SCHEMBL1958924 0.77 ATXN2 (0.42) ATXN2FFAR2BRD4CDK2CDK1
SCHEMBL15067934 0.75 BRD4 (0.47) FFAR2BRD4CDK2CDK1CCNB1
SCHEMBL1808876 0.74 GRM4 (0.42) ALDH1A1GRM4
SCHEMBL15067526 0.74 BRD4 (0.52) ATXN2FFAR2BRD4GRM4
SCHEMBL1699966 0.72 CA1 (0.58) ALDH1A1PIK3CDPIK3CBPIK3CG
SCHEMBL1700813 0.72 XDH (0.38) ATXN2BRD4
SCHEMBL1699938 0.70 BCL2 (0.39) BRD4ALDH1A1PIK3CDPIK3CG
SCHEMBL1958468 0.70 FFAR2 (0.42) ATXN2FFAR2BRD4GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109897038-B Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases 艾伯维爱尔兰无限公司 2022-04-05 CN disclosed
CN-108175749-B Melt-extruded solid dispersions containing apoptosis-inducing agents 艾伯维爱尔兰无限公司 2021-09-10 CN disclosed