SCHEMBL8322680

SCHEMBL8322680

N#Cc1ccc(N(Cc2ccc(Cl)c(Cl)c2)c2cncnc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 17/20 0.45
STS P08842 1/20 0.39
PYCR1 P32322 1/20 0.36
NR1I3 Q14994 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328066 0.86 CYP19A1 (0.44) CYP19A1STS
SCHEMBL8329428 0.85 MAOA (0.42) CYP19A1
SCHEMBL8327043 0.82 CYP19A1 (0.45) CYP19A1STS
SCHEMBL8326433 0.80 CYP19A1 (0.39) CYP19A1STS
SCHEMBL8325528 0.80 CYP19A1 (0.53) CYP19A1
SCHEMBL8323103 0.80 ESR1 (0.49) CYP19A1
SCHEMBL8329139 0.80 KCNJ1 (0.49) CYP19A1
SCHEMBL28922397 0.80 CYP19A1 (0.46) CYP19A1STS
SCHEMBL8324221 0.80 AR (0.45) CYP19A1
SCHEMBL8329384 0.79 CYP19A1 (0.43) CYP19A1STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed