SCHEMBL28923911

SCHEMBL28923911

CCOC(=O)C(=O)Cc1ccc(F)c(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.48
TSHR P16473 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CNR2 P34972 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
LMNA P02545 2/20 0.41
HTT P42858 1/20 0.41
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
KCNJ6 P48051 1/20 0.40
KCNJ5 P48544 1/20 0.40
KCNJ3 P48549 1/20 0.40
ABCB1 P08183 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7640320 0.86 TSHR (0.57) PIK3CATSHRSMN1; SMN2ALDH1A1MAPT
SCHEMBL7641749 0.86 ALDH1A1 (0.48) TSHRALDH1A1MAPTMEN1KMT2A
SCHEMBL28923912 0.83 PIK3CA (0.44) PIK3CATSHRSMN1; SMN2ALDH1A1MAPT
SCHEMBL23049584 0.82 MEN1 (0.43) TSHRSMN1; SMN2ALDH1A1MAPTALOX15
SCHEMBL5808567 0.81 MAPT (0.52) TSHRSMN1; SMN2ALDH1A1MAPTALOX15
SCHEMBL30965434 0.79 TSHR (0.57) TSHRSMN1; SMN2ALDH1A1MAPTMEN1
SCHEMBL20681282 0.79 TSHR (0.57) TSHRSMN1; SMN2ALDH1A1MAPTMEN1
SCHEMBL5792784 0.79 MAPT (0.49) PIK3CASMN1; SMN2ALDH1A1MAPTMEN1
SCHEMBL1699588 0.78 PIK3CA (0.44) PIK3CATSHRSMN1; SMN2ALDH1A1MAPT
SCHEMBL1699591 0.78 PIK3CA (0.44) PIK3CATSHRSMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109761986-B Tricyclic derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2021-10-08 CN disclosed