SCHEMBL28923975

SCHEMBL28923975

NC(=O)Oc1ccc(N2CCN(c3ccc(O)cc3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.55
GAA P10253 6/20 0.55
KDM4E B2RXH2 4/20 0.55
ALDH1A1 P00352 4/20 0.55
USP2 O75604 2/20 0.55
KMT2A Q03164 2/20 0.55
LMNA P02545 2/20 0.50
TDP1 Q9NUW8 1/20 0.49
ME2 P23368 6/20 0.48
ME1 P48163 6/20 0.48
ME3 Q16798 6/20 0.48
PKM P14618 1/20 0.46
NPC1 O15118 1/20 0.46
ALOX15 P16050 2/20 0.44
ITGB3 P05106 2/20 0.44
ITGA2B P08514 2/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HSD17B10 Q99714 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542788 0.86 ALDH1A1 (0.47) MAPTGAAKDM4EALDH1A1USP2
SCHEMBL28106920 0.85 GAA (0.56) MAPTGAAKDM4EALDH1A1KMT2A
SCHEMBL28304654 0.85 L3MBTL1 (0.62) MAPTGAAKDM4EALDH1A1KMT2A
SCHEMBL20640028 0.85 MAPT (0.50) MAPTGAAALDH1A1USP2KMT2A
SCHEMBL28096400 0.84 ALDH1A1 (0.50) MAPTGAAKDM4EALDH1A1USP2
Hydrochloric Acid SCHEMBL10436132 0.83 L3MBTL1 (0.60) MAPTGAAKDM4EALDH1A1KMT2A
SCHEMBL348122 0.83 MEN1 (0.54) MAPTGAAKDM4EKMT2ALMNA
SCHEMBL3914229 0.83 AKR1C3 (0.51) MAPTGAAKDM4EALDH1A1KMT2A
SCHEMBL29771394 0.82 GFER (0.51) MAPTGAAKDM4EALDH1A1USP2
SCHEMBL27922475 0.79 KDM4E (0.52) MAPTGAAKDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115536602-A Preparation method of posaconazole intermediate 成都海博为药业有限公司 2022-12-30 CN claimed
CN-114594192-A Method for detecting chloroaniline and chloronitroaniline isomers in posaconazole starting material 山东大学 2022-06-07 CN claimed
CN-115536602-A Preparation method of posaconazole intermediate 成都海博为药业有限公司 2022-12-30 CN disclosed
CN-114594192-A Method for detecting chloroaniline and chloronitroaniline isomers in posaconazole starting material 山东大学 2022-06-07 CN disclosed