SCHEMBL28924972

SCHEMBL28924972

Cn1cc(Oc2ccc(S(C)(=O)=O)cc2)c(-c2cccc3[nH]ncc23)n1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.60
PIK3CD O00329 2/20 0.60
PIK3CB P42338 1/20 0.60
PIK3CG P48736 1/20 0.60
PRKDC P78527 1/20 0.60
BRAF P15056 3/20 0.48
CYP11B1 P15538 2/20 0.42
CYP11B2 P19099 2/20 0.42
METAP2 P50579 2/20 0.40
PTK6 Q13882 1/20 0.40
RAF1 P04049 2/20 0.38
CREBBP Q92793 1/20 0.38
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
PTGS2 P35354 1/20 0.38
BRD4 O60885 2/20 0.38
GCK P35557 1/20 0.38
MAPK8 P45983 1/20 0.36
PIK3R1 P27986 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28640313 0.84 PIK3CA (0.59) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL28631330 0.80 BRAF (0.56) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL28635804 0.80 BRAF (0.51) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL28924973 0.76 PIK3CA (0.56) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL561236 0.75 PIK3CA (1.00) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL28961950 0.73 BRAF (0.61) PIK3CABRAFMETAP2RAF1CREBBP
SCHEMBL2195217 0.72 PIK3CA (1.00) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL17739228 0.70 CYP11B1 (0.55) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC
SCHEMBL22886577 0.70 BRAF (0.57) PIK3CABRAFMETAP2CREBBPBRD4
SCHEMBL28640314 0.69 PIK3CA (0.52) PIK3CAPIK3CDPIK3CBPIK3CGPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106659765-B Use of dianhydrogalactitol and analogs or derivatives thereof for treating non-small cell lung cancer and ovarian cancer 德玛医药 2021-08-13 CN disclosed