SCHEMBL28640314

SCHEMBL28640314

Cn1cc(-c2ccc(S(C)(=O)=O)cc2-c2cccc3[nH]ncc23)cn1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.52
METAP2 P50579 3/20 0.49
PIK3CD O00329 1/20 0.48
PIK3CB P42338 1/20 0.48
PIK3CG P48736 1/20 0.48
PRKDC P78527 1/20 0.48
BRAF P15056 3/20 0.45
KCNH2 Q12809 1/20 0.41
RAF1 P04049 2/20 0.41
LRRK2 Q5S007 1/20 0.41
BRD4 O60885 3/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TTK P33981 1/20 0.39
MAPK8 P45983 1/20 0.39
LOXL2 Q9Y4K0 2/20 0.39
LOX P28300 1/20 0.39
PTK6 Q13882 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28924973 0.82 PIK3CA (0.56) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL3433766 0.81 METAP2 (0.51) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL3435046 0.78 BRD4 (0.56) PIK3CAMETAP2BRAFRAF1BRD4
SCHEMBL28640313 0.75 PIK3CA (0.59) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL3435505 0.74 METAP2 (0.48) PIK3CAMETAP2BRAFLRRK2BRD4
SCHEMBL561550 0.70 PIK3CA (0.75) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL2193765 0.69 PIK3CA (0.82) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL28924972 0.69 PIK3CA (0.60) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL2194222 0.68 PIK3CA (1.00) PIK3CAMETAP2PIK3CDPIK3CBPIK3CG
SCHEMBL17739226 0.67 METAP2 (0.62) METAP2BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106659765-B Use of dianhydrogalactitol and analogs or derivatives thereof for treating non-small cell lung cancer and ovarian cancer 德玛医药 2021-08-13 CN disclosed