SCHEMBL28924976

SCHEMBL28924976

C=CC(=O)Oc1ccccc1OCc1ccc(F)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.52
RAB9A P51151 1/20 0.52
LMNA P02545 3/20 0.51
MAPT P10636 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
NPC1 O15118 1/20 0.48
ALDH1A1 P00352 3/20 0.47
HPGD P15428 1/20 0.47
PLA2G1B P04054 1/20 0.46
ATG4B Q9Y4P1 1/20 0.46
KDM4E B2RXH2 1/20 0.46
AKR1C3 P42330 1/20 0.46
RXRA P19793 2/20 0.45
RXRB P28702 1/20 0.45
RXRG P48443 1/20 0.45
MEN1 O00255 1/20 0.44
SLC1A5 Q15758 1/20 0.44
PTPRC P08575 1/20 0.44
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6026935 0.89 NPC1 (0.51) MAPTL3MBTL1NPC1RXRATHRA
SCHEMBL21647816 0.85 LRRK2 (0.47) LMNAMAPTL3MBTL1NPC1ALDH1A1
SCHEMBL29413361 0.79 THRB (0.56) KMT2AMAPTALDH1A1HPGDKDM4E
SCHEMBL3841280 0.79 THRB (0.56) KMT2AMAPTALDH1A1HPGDKDM4E
SCHEMBL27849251 0.78 NPC1 (0.53) KMT2ALMNAMAPTL3MBTL1NPC1
SCHEMBL7104109 0.77 THRB (0.51) KMT2ALMNAMAPTL3MBTL1NPC1
SCHEMBL10717803 0.77 L3MBTL1 (0.50) RAB9ALMNAMAPTL3MBTL1NPC1
SCHEMBL819105 0.76 THRB (0.56) LMNAMAPTL3MBTL1ALDH1A1THRA
SCHEMBL30197447 0.76 THRB (0.56) LMNAMAPTL3MBTL1ALDH1A1THRA
SCHEMBL28820774 0.76 ABCB1 (0.54) MAPTAKR1C3SLC1A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109153636-B Cyclopropyl-amide compounds as dual LSD1/HDAC inhibitors 朱比连特埃皮科尔有限责任公司 2021-10-22 CN disclosed