SCHEMBL28926323

SCHEMBL28926323

C[C@@H](Cc1cc(C#N)c2c(c1)CCN2CCCOC(=O)c1ccccc1)NCCOc1ccccc1OCC(F)(F)F

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 20/20 0.64
ADRA1D P25100 19/20 0.64
ADRA1B P35368 19/20 0.64
HTR1A P08908 2/20 0.64
ADRA2A P08913 2/20 0.64
ADRA2B P18089 2/20 0.64
ADRA2C P18825 2/20 0.64
HRH1 P35367 2/20 0.64
OPRM1 P35372 2/20 0.64
DRD3 P35462 2/20 0.64
HTR2B P41595 2/20 0.64
SLC6A3 Q01959 2/20 0.64
KCNH2 Q12809 2/20 0.64
ADRB2 P07550 1/20 0.64
DRD2 P14416 1/20 0.64
DRD1 P21728 1/20 0.64
DRD4 P21917 1/20 0.64
PTGS1 P23219 1/20 0.64
HTR1D P28221 1/20 0.64
HTR1B P28222 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13729913 1.00 ADRA1A (0.64) ADRA1AADRA1DADRA1BHTR1AADRA2A
SCHEMBL524564 1.00 ADRA1A (0.64) ADRA1AADRA1DADRA1BHTR1AADRA2A
Oxalic Acid SCHEMBL526172 0.99 ADRA1A (0.62) ADRA1AADRA1DADRA1BHTR1AADRA2A
Oxalic Acid SCHEMBL28644141 0.99 ADRA1A (0.62) ADRA1AADRA1DADRA1BHTR1AADRA2A
Oxalic Acid SCHEMBL28644138 0.99 ADRA1A (0.62) ADRA1AADRA1DADRA1BHTR1AADRA2A
SCHEMBL18157802 0.96 ADRA1D (0.62) ADRA1AADRA1DADRA1BHTR1AADRA2A
Alpha-Ketoglutaric Acid SCHEMBL17026691 0.94 ADRA1D (0.58) ADRA1AADRA1DADRA1BHTR1AADRA2A
SCHEMBL13037438 0.92 ADRA1A (0.59) ADRA1AADRA1DADRA1BHTR1AADRA2A
SCHEMBL28996811 0.92 ADRA1D (0.66) ADRA1AADRA1DADRA1BHTR1AADRA2A
SCHEMBL19730677 0.92 ADRA1D (0.55) ADRA1AADRA1DADRA1BHTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110452149-B Preparation method of indoline compound, indoline compound and application 北京鑫开元医药科技有限公司 2021-11-02 CN disclosed