SCHEMBL289322

SCHEMBL289322

Cc1nc(-c2ccc(-c3cccnc3)s2)sc1CC=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 12/20 0.48
CYP2C19 P33261 9/20 0.48
CYP3A4 P08684 8/20 0.48
CYP2C9 P11712 7/20 0.48
CYP2E1 P05181 6/20 0.48
CYP2B6 P20813 5/20 0.48
CYP2D6 P10635 6/20 0.45
CYP1A2 P05177 2/20 0.44
LMNA P02545 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
MAPT P10636 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL289748 0.99 CYP2A6 (0.47) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
SCHEMBL1679708 0.90 CYP3A4 (0.54) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
SCHEMBL289268 0.77 KDM4E (0.46) LMNAMAPTHDAC1KDM4E
SCHEMBL851867 0.77 SMN1; SMN2 (0.51) LMNAMAPTKDM4E
SCHEMBL289321 0.74 CYP3A4 (0.62) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
SCHEMBL289879 0.74 CYP3A4 (0.62) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
SCHEMBL29828863 0.74 CYP3A4 (0.58) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
SCHEMBL6513272 0.74 CYP2A6 (0.67) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
Hydrochloric Acid SCHEMBL289747 0.73 CYP3A4 (0.61) CYP2A6CYP2C19CYP3A4CYP2C9CYP2E1
SCHEMBL288142 0.73 KDM4E (0.54) LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed