SCHEMBL289879

SCHEMBL289879

Cc1nc(-c2ccc(-c3cccnc3)s2)sc1C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.62
CYP2C19 P33261 5/20 0.62
CYP1A2 P05177 4/20 0.62
LMNA P02545 1/20 0.62
SMN1; SMN2 Q16637 3/20 0.61
MKNK1 Q9BUB5 1/20 0.56
MKNK2 Q9HBH9 1/20 0.56
KDM4E B2RXH2 5/20 0.56
RAB9A P51151 3/20 0.52
GAA P10253 1/20 0.52
KMT2A Q03164 4/20 0.52
CYP2C9 P11712 3/20 0.52
MEN1 O00255 3/20 0.52
CYP2D6 P10635 2/20 0.52
CYP2A6 P11509 2/20 0.51
GPR35 Q9HC97 1/20 0.50
NPC1 O15118 1/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 2/20 0.49
ALDH1A1 P00352 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289321 0.90 CYP3A4 (0.62) CYP3A4CYP2C19CYP1A2LMNASMN1; SMN2
SCHEMBL595294 0.89 CYP1A2 (0.77) CYP3A4CYP2C19CYP1A2LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL289747 0.88 CYP3A4 (0.61) CYP3A4CYP2C19CYP1A2LMNASMN1; SMN2
Hydrochloric Acid SCHEMBL11388179 0.88 CYP1A2 (0.75) CYP3A4CYP2C19CYP1A2LMNASMN1; SMN2
SCHEMBL289596 0.88 SMN1; SMN2 (0.74) LMNASMN1; SMN2KDM4ERAB9AGAA
SCHEMBL2785654 0.87 CYP3A4 (0.60) CYP3A4CYP2C19CYP1A2LMNASMN1; SMN2
SCHEMBL289408 0.86 SMN1; SMN2 (0.72) LMNASMN1; SMN2KDM4ERAB9AGAA
SCHEMBL289784 0.84 CDC7 (0.62) CYP3A4CYP2C19CYP1A2LMNAKDM4E
Hydrochloric Acid SCHEMBL289783 0.83 CDC7 (0.61) CYP3A4CYP2C19CYP1A2LMNAKDM4E
SCHEMBL290134 0.81 KDM4E (0.75) LMNASMN1; SMN2KDM4ERAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427447-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION Pike Pharma GmbH (CH) 2012-03-14 EP disclosed
WO-2010128163-A2 SMALL MOLECULE INHIBITORS OF INFLUENZA A AND B VIRUS AND RESPIRATORY SYNCYTIAL VIRUS REPLICATION PIKE PHARMA GMBH (CH) 2010-11-11 WO disclosed