SCHEMBL28934476

SCHEMBL28934476

CCOCOc1cc(C#N)ccc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.41
DRD4 P21917 1/20 0.32
TDP2 O95551 2/20 0.31
S1PR1 P21453 1/20 0.31
NR3C2 P08235 3/20 0.30
NR3C1 P04150 2/20 0.30
PGR P06401 2/20 0.30
AR P10275 2/20 0.30
ESR2 Q92731 1/20 0.30
LPL P06858 1/20 0.30
LIPG Q9Y5X9 1/20 0.30
PDE4B Q07343 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30101076 1.00 TRPV4 (0.41) TRPV4DRD4TDP2S1PR1NR3C2
SCHEMBL22323989 0.88 TRPV4 (0.36) TRPV4TDP2ARESR2PDE4B
SCHEMBL29447080 0.88 TRPV4 (0.36) TRPV4TDP2ARESR2PDE4B
SCHEMBL25260899 0.87 EGFR (0.30) LPLLIPG
SCHEMBL30936689 0.85 TRPV4 (0.33) TRPV4
SCHEMBL25859550 0.83
SCHEMBL28691150 0.82 TRPV4 (0.33) TRPV4
SCHEMBL25300289 0.81 CHRNB2 (0.33)
SCHEMBL4141794 0.81 AR (0.42) TRPV4ARPDE4B
SCHEMBL28934910 0.81 UCHL1 (0.39) LPLLIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116410140-A NLRP3 inflammation corpuscle inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2023-07-11 CN disclosed
CN-115433163-A NLRP3 inflammasome inhibitor and application thereof 药捷安康(南京)科技股份有限公司 2022-12-06 CN disclosed